Xanomeline Tartrate
Product Sizes
10 mg
£169.00
SIH-642-10MG
50 mg
£400.00
SIH-642-50MG
About this Product
- SKU:
- SIH-642
- Additional Names:
- 3-[4-(Hexyloxy)-1,2,5-thiadiazol-3-yl]-1,2,5,6-tetrahydro-1-methylpyridine, tartrate, LY-246708; NNC-11-0232
- CAS Number:
- 152854-19-8
- CE/IVD:
- Not for use in humans. Not for use in diagnostics or therapeutics. For in vitro research use only.
- Extra Details:
- A functionally selective M1 muscarinic receptor agonist with high affinity for central muscarinic subtypes (EC₅₀ = 0.3, 92.5, 5, 52, and 42 nM for M1, M2, M3, M4, and M5, respectively). Its strong selectivity for M1 receptors underlies a range of central nervous system effects, including positive cognitive and behavioral improvements in models of schizophrenia and Alzheimer's disease. Beyond its neurocognitive actions, the compound also suppresses pro-inflammatory cytokine responses and enhances survival in sepsis models. Additionally, it demonstrates potent analgesic efficacy in rodent models of chronic inflammatory and neuropathic pain, indicating broad therapeutic potential across neuroimmune and pain-processing pathways.
- Molecular Weight:
- 431.5
- Purity:
- >98%
- Shipping Conditions:
- Ambient
- Source:
- Synthetic
- Storage Conditions:
- -20[o]C
- Supplier:
- StressMarq Biosciences
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Manufacturer's Data Sheet:https://www.stressmarq.com/products/small-molecules/agonist/xanomeline-tartrate-sih-642/
