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Proteins and Peptides

(E)-3;4;5-Trimethoxycinnamic acid

Product Sizes
100 mg
£ POA
HY-W050162-100MG
50 mg
£ POA
HY-W050162-50MG
1 g
£ POA
HY-W050162-1G
500 mg
£ POA
HY-W050162-500MG
10mM/1mL
£ POA
HY-W050162-10MM
About this Product
SKU:
HY-W050162
Additional Names:
TMCA
CAS Number:
20329-98-0
Extra Details:
(E)-3;4;5-Trimethoxycinnamic acid (TMCA) is a cinnamic acid substituted by multi-methoxy groups. (E)-3;4;5-Trimethoxycinnamic acid is an orally active and potent GABAA/BZ receptor agonist. (E)-3;4;5-Trimethoxycinnamic exhibits favourable binding affinity to 5-HT2C and 5-HT1A receptor; with IC50 values of 2.5 and 7.6 μM; respectively. (E)-3;4;5-Trimethoxycinnamic acid shows anticonvulsant and sedative activity. (E)-3;4;5-Trimethoxycinnamic acid can be used for the research of insomnia; headache and epilepsy[1][2][3].
Molecular Weight:
238.24
Purity:
99.97
References:
[1]Zhao Z, et al. Research progress in the biological activities of 3,4,5-trimethoxycinnamic acid (TMCA) derivatives. Eur J Med Chem. 2019 Jul 1;173:213-227.|[2]Chen CY, et al. 3,4,5-Trimethoxycinnamic acid, one of the constituents of Polygalae Radix exerts anti-seizure effects by modulating GABAAergic systems in mice. J Pharmacol Sci. 2016 May;131(1):1-5. |[3]Lee CI, et al. 3,4,5-Trimethoxycinnamic acid (TMCA), one of the constituents of Polygalae Radix enhances pentobarbital-induced sleeping behaviors via GABAAergic systems in mice. Arch Pharm Res. 2013 Oct;36(10):1244-51.
Research Area:
Neurological Disease
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C; 3 years; 4[o]C; 2 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
GPCR/G Protein;Membrane Transporter/Ion Channel;Neuronal Signaling
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