Anrikefon (acetate)
Product Sizes
10 mg
£ POA
HY-P3445A-10MG
5 mg
£ POA
HY-P3445A-5MG
1 mg
£ POA
HY-P3445A-1MG
About this Product
- SKU:
- HY-P3445A
- Additional Names:
- HSK21542 (acetate)
- CAS Number:
- 2584931-05-3
- Extra Details:
- Anrikefon (HSK21542) acetate is a peripherally restricted κ-opioid receptor (KOR) agonist with an IC50 of 0.54 nM; an EC50 of 2.41 pM; and a Kₐ of 0.068 nM against human KOR; and it shows high selectivity over μ and δ opioid receptors. Anrikefon exerts analgesic effects by inhibiting behavioral responses associated with inflammatory; postoperative and neuropathic pain; and also exerts antipruritic effects by reducing itch-related behaviors. Anrikefon acetate can be used in the research of pain; pruritus; and pruritus associated with chronic kidney disease[1][2].
- Molecular Weight:
- 763.97
- Purity:
- 99.68
- References:
- [1]WHO Drug Information, Vol. 36, No. 2, 2022. Geneva: World Health Organization; 2022. Licence: CC BY-NC-SA 3.0 IGO.
- Research Area:
- Neurological Disease
- Shipping Conditions:
- Blue Ice
- Storage Conditions:
- -80[o]C; 2 years; -20[o]C; 1 year (Powder; sealed storage; away from moisture)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Peptides
- Pathway:
- GPCR/G Protein;Neuronal Signaling
