Anrikefon
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HY-P3445-1EACH
About this Product
- SKU:
- HY-P3445
- Additional Names:
- HSK21542
- CAS Number:
- 2269511-95-5
- Extra Details:
- Anrikefon is a peripherally restricted kappa opioid receptor (KOR) agonist; with an IC50 of 0.54 nM; an EC50 of 2.41 pM; and a Ka of 0.068 nM against human KOR; and it exhibits high selectivity over μ and δ opioid receptors. Anrikefon exerts analgesic effects by inhibiting behaviors associated with inflammatory; postoperative and neuropathic pain; and also exerts antipruritic effects by reducing itch-related behaviors. Anrikefon can be used in research on pain; pruritus; and pruritus associated with chronic kidney disease[1][2].
- Molecular Weight:
- 703.91
- References:
- [1]WHO Drug Information, Vol. 36, No. 2, 2022. Geneva: World Health Organization; 2022. Licence: CC BY-NC-SA 3.0 IGO.
- Research Area:
- Neurological Disease
- Shipping Conditions:
- Ambient
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Peptides
