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Proteins and Peptides

7ACC2

Product Sizes
5 mg
£ POA
HY-D0713-5MG
2 mg
£ POA
HY-D0713-2MG
100 mg
£ POA
HY-D0713-100MG
10 mg
£ POA
HY-D0713-10MG
50 mg
£ POA
HY-D0713-50MG
25 mg
£ POA
HY-D0713-25MG
10mM/1mL
£ POA
HY-D0713-10MM
About this Product
SKU:
HY-D0713
Application:
Antibody Microarray
CAS Number:
1472624-85-3
Extra Details:
7ACC2 is a potent monocarboxylate transporter (MCT) inhibitor with an IC50 of 11 nM for inhibition of [14C]-lactate influx. 7ACC2 is also a potent inhibitor of mitochondrial pyruvate transport. 7ACC2 is an anticancer agent through inhibition of lactate flux[1][2].
Molecular Weight:
309.32
Purity:
99.95
References:
[1]Draoui N, et al. Synthesis and pharmacological evaluation of carboxycoumarins as a new antitumor treatment targeting lactate transport in cancer cells. Bioorg Med Chem. 2013 Nov 15;21(22):7107-17.|[2]Cyril Corbet, et al. Interruption of lactate uptake by inhibiting mitochondrial pyruvate transport unravels direct antitumor and radiosensitizing effects. Nat Commun. 2018 Mar 23;9(1):1208.
Research Area:
Cancer
Shipping Conditions:
Ambient
Storage Conditions:
4[o]C (Powder; protect from light)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Fluorophores
Pathway:
Membrane Transporter/Ion Channel;Metabolic Enzyme/Protease
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