Pimethixene
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HY-B1101-1EACH
About this Product
- SKU:
- HY-B1101
- Additional Names:
- Pimetixene
- Application:
- Electron Microscopy
- CAS Number:
- 314-03-4
- Extra Details:
- Pimethixene is antihistamine and antiserotonergic compound; acts as an antimigraine agent. Pimethixene is a highly potent antagonist of 5-HT1A; 5-HT2A; 5-HT2B; 5-HT2C; histamine H1; dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors; with pKis of 7.63; 10.22; 10.44; 8.42; 10.14; 8.19; 7.54; 8.61 and 9.38; respectively[1].
- Molecular Weight:
- 293.43
- References:
- [1]Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80.
- Research Area:
- Neurological Disease; Endocrinology
- Shipping Conditions:
- Ambient
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
