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Proteins and Peptides

AZ-5104

Product Sizes
100 mg
£ POA
HY-B0793-100MG
10 mg
£ POA
HY-B0793-10MG
50 mg
£ POA
HY-B0793-50MG
200 mg
£ POA
HY-B0793-200MG
5 mg
£ POA
HY-B0793-5MG
10mM/1mL
£ POA
HY-B0793-10MM
25 mg
£ POA
HY-B0793-25MG
About this Product
SKU:
HY-B0793
CAS Number:
1421373-98-9
Extra Details:
AZ-5104 is an active; demethylated metabolite of AZD 9291. AZ-5104 is an EGFR inhibitor with IC50s of 1; 6; 1; 25 and 7 nM for EGFRL858R/T790M; EGFRL858R; EGFRL861Q; EGFR and ErbB4; respectively.
Molecular Weight:
485.58
Purity:
99.91
References:
[1]Cross DA, et al. AZD9291, an irreversible EGFR TKI, overcomes T790M-mediated resistance to EGFR inhibitors in lung cancer. Cancer Discov. 2014 Sep;4(9):1046-61.
Research Area:
Cancer
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C; 3 years; 4[o]C; 2 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
JAK/STAT Signaling;Protein Tyrosine Kinase/RTK
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