Skip to content

Basket

You currently have no items in your basket.

Total (excl. vat) £0.00
View basket & checkout
Proteins and Peptides

BE2012

Product Sizes
50 mg
£ POA
HY-180944-50MG
5 mg
£ POA
HY-180944-5MG
10 mg
£ POA
HY-180944-10MG
25 mg
£ POA
HY-180944-25MG
100 mg
£ POA
HY-180944-100MG
10mM/1mL
£ POA
HY-180944-10MM
About this Product
SKU:
HY-180944
CAS Number:
667889-47-6
Extra Details:
BE2012; SR8278 (HY-14415) derivative; is a potent and selective REV-ERBα/β Antagonist with EC50 values of 0.285 and 0.346 μM. BE2012 binds to the ligand-binding domain (LBD) of REV-ERB; preventing the receptor from recruiting co-inhibitory factors and thereby releasing the transcriptional repression on downstream target genes. BE2012 can upregulate the expression of myogenic transcription factors Myf5 and Myod; promoting muscle regeneration and repair in acute muscle injury micemodels[1].
Molecular Weight:
293.36
Purity:
99.49
Research Area:
Neurological Disease
Shipping Conditions:
Ambient
Storage Conditions:
4[o]C (Powder; stored under nitrogen)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Price enquiry form