(E)-Belizatinib
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HY-17603A-1EACH
About this Product
- SKU:
- HY-17603A
- Additional Names:
- (E)-TSR-011
- CAS Number:
- 1388225-72-6
- Extra Details:
- (E)-Belizatinib ((E)-TSR-011)) (compound 36); the (E)-isomer of Belizatinib (HY-17603); is a potent; selective and orally active anaplastic lymphoma kinase (ALK) Inhibitor with an enzymatic IC50 of 0.005 μM and a cellular IC50 of 0.048 μM. (E)-Belizatinib shows >61-fold selectivity over JAK2; SRC; and IGF1R. (E)-Belizatinib shows favorable potency and PK characteristics in rats and dogs. (E)-Belizatinib can be used for ALK-driven cancer research[1].
- Molecular Weight:
- 577.73
- Research Area:
- Cancer
- Shipping Conditions:
- Ambient
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
