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Proteins and Peptides

BuChE-IN-10

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HY-162277-1EACH
About this Product
SKU:
HY-162277
Extra Details:
BuChE-IN-10 (compound 7p) is an inhibitor of BuChE (eqBuChE IC50 = 4.68 nM; huBuChE IC50 = 9.12 nM). BuChE-IN-10 has anti-neuroinflammatory activity and exhibits high BBB permeability[1].
Molecular Weight:
369.41
References:
[1]Chuanyu Yu, et al. Novel anti-neuroinflammatory pyranone-carbamate derivatives as selective butyrylcholinesterase inhibitors for treating Chuanyu Yu, et al. Novel anti-neuroinflammatory pyranone-carbamate derivatives as selective butyrylcholinesterase inhibitors for treating Alzheimer's disease. J Enzyme Inhib Med Chem. 2024, 39, 1.disease. J Enzyme Inhib Med Chem. 2024, 39, 1.
Research Area:
Neurological Disease
Shipping Conditions:
Ambient
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
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