(4′R)-TGR5 Receptor Agonist 4
Product Sizes
1 mg
£ POA
HY-156830A-1MG
25 mg
£ POA
HY-156830A-25MG
50 mg
£ POA
HY-156830A-50MG
5 mg
£ POA
HY-156830A-5MG
10 mg
£ POA
HY-156830A-10MG
10mM/1mL
£ POA
HY-156830A-10MM
About this Product
- SKU:
- HY-156830A
- Application:
- Electron Microscopy
- CAS Number:
- 1872436-55-9
- Extra Details:
- (4′R)-TGR5 Receptor Agonist 4 is the R enantiomer of TGR5 Receptor Agonist 4 (HY-156830). TGR5 Receptor Agonist 4 is an agonist of Bile Acid Receptor (TGR5); with EC50 for hTGR5 and mTGR5 of 2 nM and 3 nM; respectively. TGR5 Receptor Agonist 4 plays important roles in hypoglycemic and weight loss[1].
- Molecular Weight:
- 470.95
- Purity:
- 99.90
- References:
- [1]Sylvain Picon, et al. Discovery, Structure-Activity Relationships, and In Vivo Activity of Dihydropyridone Agonists of the Bile Acid Receptor TGR5. J Med Chem. 2023 Sep 14;66(17):11732-11760.
- Research Area:
- Metabolic Disease
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C; 3 years; 4[o]C; 2 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein
