(Rac)-GDC-2992
Product Sizes
1 mg
£ POA
HY-156751-1MG
5 mg
£ POA
HY-156751-5MG
About this Product
- SKU:
- HY-156751
- Additional Names:
- (Rac)-RO7656594; PROTAC AR Degrader-6
- Application:
- Antibody Microarray
- CAS Number:
- 2753650-84-7
- Extra Details:
- (Rac)-GDC-2992 (Compound 1) is a PROTAC androgen receptor degrader (DC50: 10 nM in VCaP cell). (Rac)-GDC-2992 blocks the process of androgen receptor transduction and also degrades the receptor itself. (Rac)-GDC-2992 can be used for prostate cancer research. Pink: AR ligand (HY-130845); Blue: E3 ligase ligand (HY-W1003189); Black: linker (HY-169975)[1].
- Molecular Weight:
- 819.39
- Purity:
- 95.00
- References:
- [1]Lu H.F, et al. 酞嗪酮类化合物及其制备方法和医药用途. China, WO2021249534 A1.2021-12-16.
- Research Area:
- Cancer
- Shipping Conditions:
- Blue Ice
- Storage Conditions:
- -20[o]C (Powder; protect from light; stored under nitrogen)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- PROTAC;Vitamin D Related/Nuclear Receptor
