AKR1C3-IN-10
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HY-155502-1EACH
About this Product
- SKU:
- HY-155502
- Application:
- Antibody Microarray
- CAS Number:
- 3028287-43-3
- Extra Details:
- AKR1C3-IN-10 (compound 5r) is a selective AKR1C3 inhibitor (IC50=51 nM). AKR1C3-IN-10 shows good activity in a prostate cancer xenograft model[1].
- Molecular Weight:
- 412.44
- References:
- [1]Maddeboina K, et al. Aldo-Keto Reductase 1C3 Inhibitor Prodrug Improves Pharmacokinetic Profile and Demonstrates In Vivo Efficacy in a Prostate Cancer Xenograft Model. J Med Chem. 2023 Jul 27;66(14):9894-9915.
- Research Area:
- Cancer
- Shipping Conditions:
- Ambient
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
