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Proteins and Peptides

(R)-(-)-Gossypol

Product Sizes
5 mg
HY-15464-5MG
10 mg
HY-15464-10MG
25 mg
HY-15464-25MG
10mM/1mL
HY-15464-10MM
About this Product
SKU:
HY-15464
Additional Names:
AT-101; R-(-)-gossypol acetic acid
Application:
Antibody Microarray
CAS Number:
90141-22-3
Extra Details:
(R)-(-)-Gossypol (AT-101) is the levorotatory isomer of a natural product Gossypol. AT-101 is determined to bind to Bcl-2; Mcl-1 and Bcl-xL proteins with Kis of 260±30 nM; 170±10 nM; and 480±40 nM; respectively.
Molecular Weight:
518.55
Purity:
99.37
References:
[1]Oliver CL, et al. In vitro effects of the BH3 mimetic, (-)-Gossypol, on head and neck squamous cell carcinoma cells. Clin Cancer Res. 2004 Nov 15;10(22):7757-63.|[2]Sun Y, et al. Apogossypolone, a nonpeptidic small molecule inhibitor targeting Bcl-2 family proteins, effectively inhibits growth of diffuse large cell lymphoma cells in vitro and in vivo. Cancer Biol Ther. 2008 Sep;7(9):1418-26.
Research Area:
Cancer
Shipping Conditions:
Ambient
Storage Conditions:
4[o]C (Powder; sealed storage; away from moisture and light)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
Apoptosis;Autophagy