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Proteins and Peptides

(S)-TNG260

Product Sizes
100 mg
£ POA
HY-153358A-100MG
5 mg
£ POA
HY-153358A-5MG
25 mg
£ POA
HY-153358A-25MG
50 mg
£ POA
HY-153358A-50MG
10 mg
£ POA
HY-153358A-10MG
10mM/1mL
£ POA
HY-153358A-10MM
About this Product
SKU:
HY-153358A
Application:
Antibody Microarray
CAS Number:
2935964-93-3
Extra Details:
(S)-TNG260 is an isomer of TNG260 (HY-153358). TNG260 is a CoREST selective deacetylase (CoreDAC) inhibitor. TNG260 inhibits HDAC1 with 10-fold selectivity over HDAC3. TNG260 causes HDAC1 inhibition and reverses anti-PD1 resistance driven by STK11 deletion. TNG260 reduces intratumoral infiltration of neutrophils. TNG260 exhibits immune-mediated cell killing.
Molecular Weight:
383.44
Purity:
99.78
References:
[1]Ahronian L, et al. TNG260, a CoREST-selective deacetylase inhibitor, reverses anti-PD1 resistance driven by loss of STK11[J]. J Immunother, 2022, 10(2): A1-A1595.
Research Area:
Cancer
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C; 3 years; 4[o]C; 2 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
Cell Cycle/DNA Damage;Epigenetics
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