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Proteins and Peptides

(S)-Sabutoclax

Product Sizes
5 mg
£ POA
HY-15191B-5MG
10 mg
£ POA
HY-15191B-10MG
10mM/1mL
£ POA
HY-15191B-10MM
About this Product
SKU:
HY-15191B
Additional Names:
(S)-BI-97C1
Application:
Antibody Microarray
CAS Number:
1228178-73-1
Extra Details:
(S)-Sabutoclax ((S)-BI-97C1); an optically pure apogossypol derivative; is pan-active inhibitor of antiapoptotic B-cell lymphoma/leukemia-2 (Bcl-2) family proteins. (S)-Sabutoclax (Compound II) inhibits the binding of BH3 peptides to Bcl-XL; Bcl-2; Mcl-1; and Bfl-1 with IC50 values of 0.31; 0.32; 0.20; and 0.62 μM; respectively. (S)-Sabutoclax also potently inhibits cell growth of human prostate cancer; lung cancer; and lymphoma cell lines with EC50 values of 0.13; 0.56; and 0.049 μM; respectively. (S)-Sabutoclax can be used for the research of apoptosis-based therapies against cancer[1].
Molecular Weight:
700.78
Purity:
98.03
References:
[1]Wei J, et al. BI-97C1, an optically pure Apogossypol derivative as pan-active inhibitor of antiapoptotic B-cell lymphoma/leukemia-2 (Bcl-2) family proteins. J Med Chem. 2010 May 27;53(10):4166-76.
Research Area:
Cancer
Shipping Conditions:
Blue Ice
Storage Conditions:
-20[o]C; 3 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
Apoptosis
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