Skip to content

Basket

You currently have no items in your basket.

Total (excl. vat) £0.00
View basket & checkout
Proteins and Peptides

S07-2010

Product Sizes
25 mg
£ POA
HY-150644-25MG
5 mg
£ POA
HY-150644-5MG
100 mg
£ POA
HY-150644-100MG
10 mg
£ POA
HY-150644-10MG
50 mg
£ POA
HY-150644-50MG
10mM/1mL
£ POA
HY-150644-10MM
About this Product
SKU:
HY-150644
Application:
Antibody Microarray
CAS Number:
1223194-71-5
Extra Details:
S07-2010 is a potent pan-AKR1C (aldo-keto reductase family 1 member C) inhibitor; with IC50 values of 0.19; 0.36; 0.47; and 0.73 μM for AKR1C3; AKR1C4; AKR1C1 and AKR1C2; respectively. S07-2010 induces apoptosis in A549/DDP cells. S07-2010 strengthens the cytotoxicity of chemotherapeutic agents in drug-resistant cells. S07-2010 significantly inhibits the proliferation of drug-resistant cells[1].
Molecular Weight:
371.45
Purity:
98.35
References:
[1]Siyu He, et al. Discovery of Novel Aldo-Keto Reductase 1C3 Inhibitors as Chemotherapeutic Potentiators for Cancer Drug Resistance. ACS Med. Chem. Lett. 2022.
Research Area:
Cancer
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C; 3 years; 4[o]C; 2 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
Metabolic Enzyme/Protease
Price enquiry form