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Proteins and Peptides

1-Naphthyl PP1

Product Sizes
5 mg
£ POA
HY-13941-5MG
100 mg
£ POA
HY-13941-100MG
50 mg
£ POA
HY-13941-50MG
25 mg
£ POA
HY-13941-25MG
10 mg
£ POA
HY-13941-10MG
10mM/1mL
£ POA
HY-13941-10MM
About this Product
SKU:
HY-13941
Additional Names:
1-NA-PP 1
CAS Number:
221243-82-9
Extra Details:
1-Naphthyl PP1 (1-NA-PP 1) is a selective inhibitor of src family kinases and Protein Kinase D. 1-Naphthyl PP1 inhibits v-Src and c-Fyn; c-Abl; CDK2 and CAMK II with IC50s of 1.0; 0.6; 0.6; 18 and 22 μM; respectively[1][2][3].
Molecular Weight:
317.39
Purity:
99.36
References:
[1]Bishop AC, et al. A chemical switch for inhibitor-sensitive alleles of any protein kinase. Nature. 2000 Sep 21;407(6802):395-401.|[2]Tandon M, et al. New pyrazolopyrimidine inhibitors of protein kinase d as potent anticancer agents for prostate cancer cells. PLoS One. 2013 Sep 23;8(9):e75601.|[3]Maiya R, et al. Selective chemical genetic inhibition of protein kinase C epsilon reduces ethanol consumption in mice. Neuropharmacology. 2016 Aug;107:40-48.
Research Area:
Cancer;Inflammation/Immunology;Neurological Disease
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C; 3 years; 4[o]C; 2 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
Apoptosis;Protein Tyrosine Kinase/RTK
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