(Rac)-PF-4136309
Product Sizes
50 mg
£ POA
HY-13245B-50MG
10 mg
£ POA
HY-13245B-10MG
100 mg
£ POA
HY-13245B-100MG
25 mg
£ POA
HY-13245B-25MG
1 mg
£ POA
HY-13245B-1MG
5 mg
£ POA
HY-13245B-5MG
About this Product
- SKU:
- HY-13245B
- Additional Names:
- (Rac)-INCB8761
- CAS Number:
- 857679-55-1
- Extra Details:
- (Rac)-PF-4136309 is an isoform of PF-4136309 (HY-13245); which is a potent; selective; and orally bioavailable CCR2 antagonist; with IC50s of 5.2 nM; 17 nM and 13 nM for human; mouse and rat CCR2.
- Molecular Weight:
- 568.59
- Purity:
- 98.0
- References:
- [1]Xue CB, et al. Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist. ACS Med. Chem. Lett., 2011, 2 (12), pp 913-918.
- Research Area:
- Inflammation/Immunology
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C; 3 years; 4[o]C; 2 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein;Immunology/Inflammation
