(s)-PF-4136309
Product Sizes
5 mg
£ POA
HY-13245A-5MG
10 mg
£ POA
HY-13245A-10MG
100 mg
£ POA
HY-13245A-100MG
50 mg
£ POA
HY-13245A-50MG
10mM/1mL
£ POA
HY-13245A-10MM
25 mg
£ POA
HY-13245A-25MG
About this Product
- SKU:
- HY-13245A
- Additional Names:
- (s)-INCB8761
- Application:
- Electron Microscopy
- CAS Number:
- 1372407-07-2
- Extra Details:
- (s)-PF-4136309 is the isomer of PF-4136309 (HY-13245); and can be used as an experimental control. PF-4136309 is a potent; selective; and orally bioavailable CCR2 antagonist; with IC50s of 5.2 nM; 17 nM and 13 nM for human; mouse and rat CCR2.
- Molecular Weight:
- 568.59
- Purity:
- 98.93
- References:
- [1]Xue CB, et al. Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist. ACS Med. Chem. Lett., 2011, 2 (12), pp 913-918.
- Research Area:
- Endocrinology; Inflammation/Immunology
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C; 3 years; 4[o]C; 2 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein;Immunology/Inflammation;Others
