CBP/p300-IN-12
Product Sizes
5 mg
£ POA
HY-132197-5MG
100 mg
£ POA
HY-132197-100MG
25 mg
£ POA
HY-132197-25MG
50 mg
£ POA
HY-132197-50MG
10 mg
£ POA
HY-132197-10MG
10mM/1mL
£ POA
HY-132197-10MM
About this Product
- SKU:
- HY-132197
- Application:
- Antibody Microarray
- CAS Number:
- 2738688-57-6
- Extra Details:
- CBP/p300-IN-12 is a potent and selective covalent histone acetyltransferases p300 (IC50 of 166 nM) and CBP inhibitor. CBP/p300-IN-12 decreases the levels of H3K27Ac of PC-3 cells (EC50 of 37 nM). CBP/p300-IN-12 forms a covalent adduct with C1450[1].
- Molecular Weight:
- 667.61
- Purity:
- 99.72
- References:
- [1]Anthony Mastracchio, et al. Discovery of a Potent and Selective Covalent p300/CBP Inhibitor. ACS Med Chem Lett. 2021 Apr 5;12(5):726-731.
- Research Area:
- Cancer
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C; 3 years; 4[o]C; 2 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- Epigenetics
