Samelisant
Product Sizes
100 mg
£ POA
HY-120124-100MG
5 mg
£ POA
HY-120124-5MG
10 mg
£ POA
HY-120124-10MG
25 mg
£ POA
HY-120124-25MG
50 mg
£ POA
HY-120124-50MG
10mM/1mL
£ POA
HY-120124-10MM
About this Product
- SKU:
- HY-120124
- Additional Names:
- SUVN-G3031
- CAS Number:
- 1394808-20-8
- Extra Details:
- Samelisant (SUVN-G3031) is a potent and selective histamine H3 receptor (H3R) inverse agonist with good brain penetration and oral bioavailability. Samelisant has a similar binding affinity towards human (hH3R; Ki=8.7 nM) and rat (rH3R;Ki=9.8 nM) H3R indicating no inter-species differences. Samelisant can be used for the research of sleep-related disorders[1].
- Molecular Weight:
- 446.41
- Purity:
- 98.04
- References:
- [1]Ramakrishna Nirogi, et al. Samelisant (SUVN-G3031), a potent, selective and orally active histamine H3 receptor inverse agonist for the potential treatment of narcolepsy: pharmacological and neurochemical characterisation. Psychopharmacology (Berl). 2021 Jun;238(6):1495-1511.
- Research Area:
- Neurological Disease
- Shipping Conditions:
- Blue Ice
- Storage Conditions:
- -20[o]C; 3 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein;Immunology/Inflammation;Neuronal Signaling
