ATM Inhibitor-10
Product Sizes
1 mg
£ POA
HY-118911-1MG
5 mg
£ POA
HY-118911-5MG
25 mg
£ POA
HY-118911-25MG
100 mg
£ POA
HY-118911-100MG
50 mg
£ POA
HY-118911-50MG
10 mg
£ POA
HY-118911-10MG
10mM/1mL
£ POA
HY-118911-10MM
About this Product
- SKU:
- HY-118911
- CAS Number:
- 1941214-06-7
- Extra Details:
- ATM Inhibitor-10 (compound 74); a 3-quinoline carboxamide; is a highly selective and orally active ATM inhibitor (IC50: 0.6 nM). ATM Inhibitor-10 has anti-tumor activity in SW620 xenograft models. ATM Inhibitor-10 is synergistic with Top I inhibitors[1].
- Molecular Weight:
- 434.47
- Purity:
- 98.7
- References:
- [1]Degorce SL, et al. Discovery of Novel 3-Quinoline Carboxamides as Potent, Selective, and Orally Bioavailable Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase. J Med Chem. 2016 Jul 14;59(13):6281-92.
- Research Area:
- cancer
- Shipping Conditions:
- Blue Ice
- Storage Conditions:
- -20[o]C; 3 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
