(Rac)-WAY-161503
Product Sizes
5 mg
£ POA
HY-103138A-5MG
10 mg
£ POA
HY-103138A-10MG
10mM/1mL
£ POA
HY-103138A-10MM
About this Product
- SKU:
- HY-103138A
- Application:
- Electron Microscopy
- CAS Number:
- 75704-24-4
- Extra Details:
- (Rac)-WAY-161503 is a potent; selective; highly affinity 5-HT2C receptor agonist with a Ki of 4 nM and an EC50 of 12 nM. (Rac)-WAY-161503 displays higher affinity for 5-HT2C than 5-HT2A and 5-HT2B receptors. (Rac)-WAY-161503 has anti-obesity and antidepressant effects[1][2].
- Molecular Weight:
- 272.13
- Purity:
- 98.49
- References:
- [1]Halberstadt AL, et al. 5-HT(2A) and 5-HT(2C) receptors exert opposing effects on locomotor activity in mice. Neuropsychopharmacology. 2009 Jul;34(8):1958-67.|[2]Welmaker GS, et al. Synthesis and 5-hydroxytryptamine (5-HT) activity of 2,3,4,4a-tetrahydro-1H-pyrazino[1,2-a]quinoxalin-5-(6H)ones and 2,3,4,4a,5,6-hexahydro-1H-pyrazino[1,2-a]quinoxalines. Bioorg Med Chem Lett. 2000 Sep 4;10(17):1991-4.
- Research Area:
- Metabolic Disease; Neurological Disease
- Shipping Conditions:
- Blue Ice
- Storage Conditions:
- -20[o]C; 3 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein;Neuronal Signaling
