(3aR)-Selitrectinib
Product Sizes
1 mg
£ POA
HY-101977B-1MG
About this Product
- SKU:
- HY-101977B
- Additional Names:
- (3aR)-LOXO-195
- CAS Number:
- 1350884-56-8
- Extra Details:
- (3aR)-Selitrectinib ((3aR)-LOXO-195) is an isform of Selitrectinib (HY-101977); which is a next-generation TRK kinase inhibitor; with IC50s of 0.6 nM and TRKA and TRKC; respectively[1].
- Molecular Weight:
- 380.42
- References:
- [1]Drilon A, et al. A Next-Generation TRK Kinase Inhibitor Overcomes Acquired Resistance to Prior TRK Kinase Inhibition in Patients with TRK Fusion-Positive Solid Tumors. Cancer Discov. 2017 Sep;7(9):963-972.
- Research Area:
- Cancer
- Shipping Conditions:
- Ambient
- Storage Conditions:
- 4[o]C (Powder; protect from light)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- Neuronal Signaling;Protein Tyrosine Kinase/RTK
