(Rac)-BMS-816336
Product Sizes
50 mg
£ POA
HY-101930A-50MG
10 mg
£ POA
HY-101930A-10MG
100 mg
£ POA
HY-101930A-100MG
5 mg
£ POA
HY-101930A-5MG
About this Product
- SKU:
- HY-101930A
- Application:
- Electron Microscopy
- CAS Number:
- 1009365-98-3
- Extra Details:
- (Rac)-BMS-816336 (Compound 6n) is a racemate of BMS-816336. (Rac)-BMS-816336 is a potent inhibitor of human and mouse 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) enzyme with IC50s of 10 nM and 68 nM; respectively. (Rac)-BMS-816336 has good metabolic stability[1].
- Molecular Weight:
- 341.44
- Purity:
- 99.91
- References:
- [1] Ye XY, et al. Discovery of Clinical Candidate 2-((2S,6S)-2-Phenyl-6-hydroxyadamantan-2-yl)-1-(3'-hydroxyazetidin-1-yl)ethanone [BMS-816336], an Orally Active Novel Selective 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor. J Med Chem. 2017 Jun 22;60(12):4932-4948.
- Research Area:
- Metabolic Disease
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C; 3 years; 4[o]C; 2 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- Metabolic Enzyme/Protease
