(+)-N-Allylnormetazocine (hydrochloride)
Product Sizes
5 mg
£ POA
HY-101376-5MG
About this Product
- SKU:
- HY-101376
- Additional Names:
- (+)-SKF 10047 (hydrochloride); (+)-N-Allyl-N-normetazocine (hydrochloride)
- CAS Number:
- 133005-41-1
- Extra Details:
- (+)-N-Allylnormetazocine ((+)-SKF 10047) hydrochloride is a benzomorphan opioid with psychotomi metic effects. (+)-N-Allylnormetazocine hydrochloride is an opioid receptor antagonist with Ki values of 300 nM and 27 μM for σ1 and σ2 opioid receptors; respectively. (+)-N-Allylnormetazocine hydrochloride can be used for the research of neurological disease[1][2].
- Molecular Weight:
- 293.83
- Purity:
- 99.6
- References:
- [1]May EL, et al. Synthesis and in vitro and in vivo activity of (-)-(1R,5R,9R)- and (+)-(1S,5S,9S)-N-alkenyl-, -N-alkynyl-, and -N-cyanoalkyl-5, 9-dimethyl-2'-hydroxy-6,7-benzomorphan homologues. J Med Chem. 2000 Dec 28;43(26):5030-6.|[2]Brady KT, et al. Stereoisomers of N-allylnormetazocine: phencyclidine-like behavioral effects in squirrel monkeys and rats. Science. 1982 Jan 8;215(4529):178-80.
- Research Area:
- Neurological Disease
- Shipping Conditions:
- Ambient
- Storage Conditions:
- 4[o]C (Powder; stored under nitrogen; away from moisture)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein;Neuronal Signaling
