(Rac)-VU 6008667
Product Sizes
25 mg
£ POA
HY-101281A-25MG
50 mg
£ POA
HY-101281A-50MG
5 mg
£ POA
HY-101281A-5MG
1 mg
£ POA
HY-101281A-1MG
10 mg
£ POA
HY-101281A-10MG
About this Product
- SKU:
- HY-101281A
- CAS Number:
- 2092917-63-8
- Extra Details:
- (Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM; pIC50= 5.75); has high CNS penetration[1].
- Molecular Weight:
- 438.85
- Purity:
- 99.85
- References:
- [1]McGowan KM et al, Continued optimization of the M5 NAM ML375: Discovery of VU6008667, an M5 NAM with high CNS penetration and a desired short half-life in rat for addiction studies. Bioorg Med Chem Lett. 2017 Mar 15;27(6):1356-1359.
- Research Area:
- Neurological Disease
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C; 3 years; 4[o]C; 2 years (Powder)
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
- Pathway:
- GPCR/G Protein;Neuronal Signaling
