(S)-Crizotinib (Standard)
Product Sizes
100 mg
£ POA
HY-100549R-100MG
10 mg
£ POA
HY-100549R-10MG
5 mg
£ POA
HY-100549R-5MG
50 mg
£ POA
HY-100549R-50MG
25 mg
£ POA
HY-100549R-25MG
About this Product
- SKU:
- HY-100549R
- CAS Number:
- 1374356-45-2
- Extra Details:
- (S)-Crizotinib (Standard) is the analytical standard of (S)-Crizotinib (HY-100549). This product is intended for research and analytical applications. (S)-Crizotinib is a potent and selective MTH1 (mutT homologue) inhibitor with an IC50 of 330 nM. (S)-Crizotinib disrupts nucleotide pool homeostasis via MTH1 inhibition; induces an increase in DNA single strand breaks; activates DNA repair in human colon carcinoma cells; and effectively suppresses tumour growth in animal models[1].
- Molecular Weight:
- 450.34
- Research Area:
- Cancer
- Shipping Conditions:
- Ambient
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
