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Proteins and Peptides

NPS-1034

Product Sizes
10 mg
£ POA
HY-100509-10MG
100 mg
£ POA
HY-100509-100MG
25 mg
£ POA
HY-100509-25MG
5 mg
£ POA
HY-100509-5MG
50 mg
£ POA
HY-100509-50MG
10mM/1mL
£ POA
HY-100509-10MM
About this Product
SKU:
HY-100509
CAS Number:
1221713-92-3
Extra Details:
NPS-1034 is a dual inhibitor of AXL and MET with IC50s of 10.3 and 48 nM; respectively.
Molecular Weight:
551.54
Purity:
98.0
References:
[1]Rho JK, et al. MET and AXL inhibitor NPS-1034 exerts efficacy against lung cancer cells resistant to EGFR kinase inhibitors because of MET or AXL activation. Cancer Res. 2014 Jan 1;74(1):253-62.|[2]Shin JS, et al. NPS-1034, a novel MET inhibitor, inhibits the activated MET receptor and its constitutively active mutants. Invest New Drugs. 2014 Jun;32(3):389-99.
Research Area:
Cancer
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C; 3 years; 4[o]C; 2 years (Powder)
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Pathway:
Apoptosis;Protein Tyrosine Kinase/RTK
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