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Product Sizes
5 mg
£151.00
10-5688-5MG
25 mg
£253.00
10-5688-25MG
About this Product
SKU:
10-5688
CAS Number:
896705-16-1
Extra Details:
A planar heterocyclic DNA intercalator that inhibits RNA polymerase I (Pol I), IC50 = 0.6 uM in U2OS cells, but not Pols II or III, blocking transcription elongation without inducing the DNA damage response.1-3 Inhibition disengages Pol I from chromatin, resulting in proteasome-dependent destruction of Pol I subunit RPA194.4 At nanomolar concentrations it also activates p53 in A375 cells.5
Immunogen:
DNA|RNA|Transcription factor
Molecular Weight:
360.42
Physical State:
Solid
Purity:
>98%
Purification:
HPLC Purified
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors
Sell Sheet 1:
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Sell Sheet 2:
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