C2230
Product Sizes
5 mg
£158.00
10-4955-5MG
25 mg
£267.00
10-4955-25MG
About this Product
- SKU:
- 10-4955
- CAS Number:
- 882243-88-1
- Extra Details:
- C2230 is a novel Cav2.2 channel blocker (IC50 = 1.3 uM @ -50 mV; 10.2 uM @ -80 mV) with a unique binding mode (no GPCR-mediated inhibition). It displays preferential binding to the inactive state of the channel. C2230 is active in both rat and human DRG neurons. Active in rat models of neuropathic pain and mouse models of osteoarthritis. C2230 does not affect somatosensation or motor and cardiac function.
- Immunogen:
- Ion channel
- Molecular Weight:
- 321.46
- Physical State:
- White to off-white waxy solid
- Purity:
- >98%
- Shipping Conditions:
- Ambient
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- Type:
- Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors
