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Product Sizes
5 mg
£149.00
10-4859-5MG
25 mg
£195.00
10-4859-25MG
About this Product
SKU:
10-4859
Additional Names:
CDK inhibitor, 4-[(2,6-Dichlorobenzoyl)amino]-N-piperidin-4-yl-1H-pyrazole-5-carboxamide hydrochloride
CAS Number:
902135-91-5
Extra Details:
AT7519 is a potent CDK inhibitor. Inhibits CDKs 1,2,4,5,6, and 9 (IC50s respectively: 210 nM, 47 nM, 100 nM, 13 nM, 170 nM, and <10 nM).1,2 Active in multiple human cancer cell lines.3-7 AT7519 has also been found to be a human RORG Gammat agonist.8
Immunogen:
Kinase|Retinoid receptor and related|Transcription factor
Molecular Weight:
418.7
Physical State:
Solid
Purity:
>98%
Purification:
HPLC Purified
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors