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Product Sizes
10 mg
£163.00
10-4765-10MG
50 mg
£281.00
10-4765-50MG
About this Product
SKU:
10-4765
CAS Number:
42521-82-4
Extra Details:
IPA-3 is a selective allosteric inhibitor of Group 1 p21-activated kinase (PAK1 IC50 = 2.5 uM)1 via covalent binding to the PAK1 regulatory domain preventing binding to the upstream activator Cdc422. IPA-3 has been shown to induce cell death in human leukemic cell lines3, significantly inhibit TGFB Beta1-induced prostate cell epithelial to mesenchymal transition4 and inhibits the growth of liver cancer cells5.
Immunogen:
Kinase
Molecular Weight:
350.45
Physical State:
Solid
Purity:
98%
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors