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Product Sizes
5 mg
£163.00
10-4511-5MG
10 mM (in 1 ml DMSO)
£163.00
10-4511-10MM(IN1MLDMSO)
25 mg
£195.00
10-4511-25MG
About this Product
SKU:
10-4511
Additional Names:
INCB 018424
CAS Number:
941678-49-5
Extra Details:
Potent and selective JAK1&2 inhibitor, IC50s=2.7, 4.5 and 322 nM forJAK1, JAK2 and JAK3 respectively.1 Blocks IL-6 signaling (IC50=281 nM) and proliferation of JAK2V617F+ Ba/F3 cells (IC50=127 nM).2 Inhibits the proinflammatory secretome of senescent cells.3 The JAK1 S646P mutant is highly sensitive to ruxolitinib.4 Clinically useful cancer chemotherapeutic.
Immunogen:
Kinase
Molecular Weight:
306.37
Physical State:
Solid
Purity:
99%
Purification:
HPLC Purified
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors