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Product Sizes
5 mg
£158.00
10-3743-5MG
25 mg
£243.00
10-3743-25MG
About this Product
SKU:
10-3743
Additional Names:
PF-06291826
CAS Number:
594839-88-0
Extra Details:
A potent and selective transthyretin (TTR) kinetic stabilizer. It binds selectively and with negative cooperativity to the two normally unoccupied thyroxine binding sites of the TTR tetramer (Kd = ~2 and ~200 nM)1. Stabilizes wild-type and mutant TTR under varying conditions in vitro (EC50=2.7-3.2 M).1 Clinically useful for the treatment of familial amyloid polyneuropathy2,3 and TTR-related cardiomyopathy4.
Immunogen:
UPR (Unfolded Protein Response)
Molecular Weight:
308.12
Physical State:
Solid
Purity:
98%
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules