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Product Sizes
5 mg
£173.00
10-2129-5MG
25 mg
£301.00
10-2129-25MG
About this Product
SKU:
10-2129
Additional Names:
CHIR258|TKI-258
CAS Number:
405169-16-6
Extra Details:
Potent kinase inhibitor. Inhibits FLT3 (IC50 = 1 nM), c-KIT (IC50 = 2 nM), FGFR (IC50 = 8 nM), VEGFR1/2/3 (IC50 = 10 nM), PDGFRB Beta (IC50 = 27 nM), and CSF-1R (IC50 = 36 nM).1 Active in cell culture and in whole animals. Selectively blocks the growth B9 cells transformed by wild type, or activated mutant FGFR3. Induces apoptosis, or sensitizes cells to induction of apoptosis by other means in a variety of cancer cell lines.
Immunogen:
Kinase
Molecular Weight:
392.43
Physical State:
Solid
Purity:
99%
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors