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Product Sizes
10 mg
£137.00
10-2125-10MG
50 mg
£195.00
10-2125-50MG
About this Product
SKU:
10-2125
Additional Names:
GOE-5549|N-acetyl-dinaline|PD-123654|Tacedinaline
CAS Number:
112522-64-2
Extra Details:
Orally active histone deacetylase (HDAC) inhibitor, IC50 = 0.9, 0.9, 1.2 and >20 uM for HDAC1, HDAC2, HDAC3 and HDAC8 respectively.1 Mediates G1 cell cycle arrest, inhibits proliferation and induces apoptosis in vitro and in vivo.2,3 Increases neuroplasticity during memory extinction.4 Protects beta cells from cytokine-induced apoptosis.4
Immunogen:
Protein deacetylase
Molecular Weight:
269.30
Physical State:
Solid
Purity:
98%
Purification:
HPLC Purified
Shipping Conditions:
Ambient
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Inhibitors