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Product Sizes
5 mg
£158.00
10-1486-5MG
25 mg
£281.00
10-1486-25MG
About this Product
SKU:
10-1486
CAS Number:
10023-54-8
Extra Details:
A novel small molecule thought to be an agonist at the glial cell line-derived neurotrophic factor (GDNF) family receptor A Alpha-1 GFRA Alpha-1. It inhibits radiolabeled GDNF binding in Neuro-2A cells in a concentration dependent manner IC50=10.4 uM. Like GDNF, it induced Ret autophosphorylation and promoted neurite outgrowth in Neuro-2A cells1. Recent studies indicate that it enhances GFRA Alpha family receptor signaling in conjunction with ligand stimulation. Effective treatment for small-fiber neuropathy in mouse models of the disease.2,3 GDNF agonists may be a new class of Parkinson's disease therapeutics.4
Molecular Weight:
750.45
Physical State:
Solid
Purity:
98%
Shipping Conditions:
Ambient
Storage Conditions:
RT
Supplier:
Focus Biomolecules
Type:
Proteins, Peptides, Small Molecules & Other Biomolecules: Small Molecules
Sell Sheet 1:
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