Loperamide Hydrochloride (mu-Opioid Receptor Agonist, Loperamide Hydrochloride, Imodium)

Size

£302.00

SKU:: 217515
Purity:: ≥99% (HPLC)
Storage Conditions:: 4°C
Supplier:: United States Biological
CAS Number:: 34552-83-5
Format:: Supplied as a white solid.
Extra Details:: A very potent and highly selective peripheral resctricted u-opioid receptor agonist (Ki = 2nM). Often used as an antidiarrheal, antipruritic, and antihyperalgesic agent. In addition, shown to improve defective post-receptor insulin signaling in skeletal muscle cells and enhance insulin sensitivity in rats. Synonyms: µ-Opioid Receptor Agonist, Loperamide Hydrochloride, Imodium CAS No: 34552-83-5 Molecular Formula: C₂₉H₃₃ClN₂O₂·HCl Solubility: DMSO or Warm EtOH Primary Target: u opioid receptor Primary Target Ki: 2nM Storage and Stability: May be stored at 4°C. For long-term storage, aliquot and store at 4°C. Do not freeze. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.