217283
CPCCOEt ((E)-Ethyl 1,1a,7,7a-tetrahydro-7-(hydroxyimino)cyclopropa[b]chromene-1a-carboxylate, mGlu1 Antagonist, CPCCOEt)
Size
£386.00
- SKU:
- 217283
- Molecular Weight:
- 247.25
- Purity:
- ~98% (HPLC)
- Storage Conditions:
- 4°C
- Supplier:
- United States Biological
- CAS Number:
- 179067-99-3
- Format:
- Supplied as a white powder.
- Extra Details:
- A potent, negative allosteric modulator selective for mGlu1 receptors (IC50 = 6.5uM). No effect on other mGlu subtype receptors and ionotropic glutamate receptors at concentrations less than 100uM. Acts by inhibiting an intramolecular interaction between the agonist-bound extracellular domain and the transmembrane domain. Widely used for studies related to peripheral pain and central pain pathways. CAS Number: 179067-99-3 Formula: C13H13NO4 Solubility: DMSO Primary Target: mGlu1 receptors Molar Mass: 247.25 Storage and Stability: May be stored at 4°C. For long-term storage, aliquot and store at 4°C. Do not freeze. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.
- Shipping Conditions:
- Blue Ice