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10-5635

Calphostin C

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£233.00

SKU:
10-5635
Additional Names:
PKF115-584|UCN-1028C
Physical State:
Dark red to light brown solid
Molecular Weight:
790.77
Purity:
98%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
121263-19-2
Immunogen:
Kinase
Extra Details:
Potent and specific inhibitor of protein kinase C (PKC, IC50 = 50 nM).1 Inhibition of PKC is light dependent2 and is competitive with the diacylglycerol / phorbol ester binding site1. Calphostin C competes with the diacylglycerol / phorbol ester binding site in other proteins such as Munc13-1.3 Reverses oxycodone-induced tolerance to respiratory depression.4
Shipping Conditions:
Ambient