Skip to content

Download Spec Sheet

download
  1. Shop all
  2. Antagonists

10-5362

CID16020046

Size

£158.00

SKU:
10-5362
Physical State:
Solid
Molecular Weight:
425.44
Purity:
>98%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
834903-43-4
Immunogen:
GPCR
Extra Details:
CID16020046 is a selective GPR55 antagonist.1 In HEK293 cells expressing GPR55, the compound behaves as an antagonist on lysophosphatidylinositol (LPI)-mediated Ca2+ release but was inactive on cells expressing CB1 and CB2. It blocks LPI-induced migration of colon cancer cells.2 It displays protective effects against oxidized LDL-induced inflammation3, mitigates advanced glycation end products-induced chondrocyte activation4, and displays anti-inflammatory effects in various cells5,6. A useful tool for studying the role of GPR55 in cellular physiology.
Shipping Conditions:
Ambient