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10-5092

Formoterol hemifumarate

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£166.00

SKU:
10-5092
Additional Names:
BD 40A
Physical State:
Solid
Molecular Weight:
402.5
Purity:
99%
Purification:
HPLC Purified
Storage Conditions:
RT
Supplier:
Focus Biomolecules
CAS Number:
43229-80-7
Immunogen:
GPCR
Extra Details:
Potent, long-acting agonist specific to B Beta2 (Ki = 7.6 nM), but not B Beta1 (Ki > 2.6 uM), adrenergic receptors in trachea (pD2 = 9.3) over atrium (pD2 = 7.0).1,2 Reduces adhesion and superoxide anion production in cultured activated eosinophils.3 Reverses cachexia in rats and mice via inhibition of the ATP-ubiquitin-dependent proteolytic system.4 Rescues LPS-induced motor function deficits and nigrostriatal dopamine loss in a rat model of Parkinson's.5 Clinically useful for respiratory diseases.
Shipping Conditions:
Ambient