10-5092
Formoterol hemifumarate

Size
£166.00
- SKU:
- 10-5092
- Additional Names:
- BD 40A
- Physical State:
- Solid
- Molecular Weight:
- 402.5
- Purity:
- 99%
- Purification:
- HPLC Purified
- Storage Conditions:
- RT
- Supplier:
- Focus Biomolecules
- CAS Number:
- 43229-80-7
- Immunogen:
- GPCR
- Extra Details:
- Potent, long-acting agonist specific to B Beta2 (Ki = 7.6 nM), but not B Beta1 (Ki > 2.6 uM), adrenergic receptors in trachea (pD2 = 9.3) over atrium (pD2 = 7.0).1,2 Reduces adhesion and superoxide anion production in cultured activated eosinophils.3 Reverses cachexia in rats and mice via inhibition of the ATP-ubiquitin-dependent proteolytic system.4 Rescues LPS-induced motor function deficits and nigrostriatal dopamine loss in a rat model of Parkinson's.5 Clinically useful for respiratory diseases.
- Shipping Conditions:
- Ambient
