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10-4906

DHP-103

Size

£173.00

SKU:
10-4906
Physical State:
Solid
Molecular Weight:
359.28
Purity:
>98%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
2775311-82-3
ABP:
No Import Docs
Immunogen:
Ion channel
Extra Details:
DHP-103 is a potent (IC50 = 6 nM) blocker of the intermediate-conductance calcium-activated potassium channel KCa3.1. It displays exquisite selectivity over calcium channels. It blocked mutant KCa3.1 channels that cause hereditary xerocytosis and reduced infarct volume, improved balance beam performance, and reduced activated microglia in a rat model of acute ischemic stroke.
Shipping Conditions:
Ambient