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10-4696

Selonsertib

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£149.00

SKU:
10-4696
Additional Names:
GS-4997
Physical State:
Solid
Molecular Weight:
445.5
Purity:
98%
Purification:
HPLC Purified
Storage Conditions:
-20[o]C
Supplier:
Focus Biomolecules
CAS Number:
1448428-04-3
Immunogen:
Cytochrome/MDR|Kinase
Extra Details:
Potent Apoptosis signal-regulating kinase 1 (ASK1) inhibitor (pIC50 = 8.3)1 found to improve metabolic parameters in nonalcoholic steatohepatitis, reduce hepatic steatosis, inflammation, and fibrosis2-4. Selonsertib suppressed the efflux function of multidrug resistance (MDR) transporters ABCB1 and ABCG2.5
Shipping Conditions:
Ambient