ABX-1431

Size

£158.00

SKU:: 10-4596
Physical State:: Solid
Molecular Weight:: 507.4
Purity:: 98%
Purification:: HPLC Purified
Storage Conditions:: -20[o]C
Supplier:: Focus Biomolecules
CAS Number:: 1446817-84-0
ABP:: No Import Docs
Immunogen:: Lipase
Extra Details:: Potent (IC50 = 14 nM in vitro, 2.2 nM in human PC3 cells) and very selective (>100-fold over hABHD6, >200-fold over hPLA2G7) inhibitor of monoacylglycerol lipase (MAGL).1 Active in a rat formalin pain test at 3mg/kg. Orally bioavailable and CNS penetrant.