10-4542
UNC1999
Size
£157.00
- SKU:
- 10-4542
- Physical State:
- Solid
- Molecular Weight:
- 569.74
- Purity:
- 98%
- Purification:
- HPLC Purified
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- CAS Number:
- 1431612-23-5
- Immunogen:
- Protein methyltransferase
- Extra Details:
- UNC1999 is an orally bioavailable, highly selective inhibitor of both wild-type and mutant EZH1 and EZH2 lysine methyltransferases (IC50's = 45 nM and 2 nM respectively).1 Inhibition of EZH2 with UNC1999 enhanced the efficacy of gefitinib in suppressing the proliferation of colon cancer cells
- Shipping Conditions:
- Ambient