10-4201
S1RA
Size
£182.00
- SKU:
- 10-4201
- Additional Names:
- E-52862 HCl
- Physical State:
- Solid
- Molecular Weight:
- 373.88
- Purity:
- 98%
- Purification:
- HPLC Purified
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- CAS Number:
- 1265917-14-3
- Immunogen:
- ER/Golgi
- Extra Details:
- S1RA (E-52862) is a potent and selective 1 antagonist with weak binding at 2 (IC50's: 1 = 17nM, 2 = 9300nM).1,2 S1RA abolished mechanical and thermal hyperalgesia in mice with carrageenan-induced acute inflammation by enhancing the action of endogenous opioid peptides of immune origin in a 1 dependent manner.3 BD1063 potentiated u-opioid antinociception in mice in a -dependent manner.4 S1RA displayed neuroprotective effects in a mouse model of ischemic stroke.5
- Shipping Conditions:
- Ambient