10-4172
GSK2636771
Size
£182.00
- SKU:
- 10-4172
- Physical State:
- Solid
- Molecular Weight:
- 433.43
- Purity:
- >98%
- Purification:
- HPLC Purified
- Storage Conditions:
- -20[o]C
- Supplier:
- Focus Biomolecules
- CAS Number:
- 1372540-25-4
- Immunogen:
- GPCR|Kinase
- Extra Details:
- GSK2636771 is a potent, selective (>1000-fold over A Alpha, 10-fold over D Delta, and >2000-fold over G Gamma), and orally bioavailable inhibitor of PI3KB Beta (IC50 = 5.2 nM).1 Active in vitro against multiple types of PTEN-deficient cancer cells. GSK2636771 potently blocked migration and invasion of DU145 prostate cancer cells.2 GSK2636771 has also been identified as a GPR39 agonist.3
- Shipping Conditions:
- Ambient